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Patents & International Journal Articles:

16. A Novel Synthesis of a Triazolesulfonyl Chloride as a Precursor for GlyT-1 Inhibitors Visweswaran Parthasarathy; Edmund Carulli; Kashinath Sadalapure; Ron Buckle; Christopher L. Cioffi; Karl E. Reineke; Shuang Liu; UK-Singapore Symposium on Contemporary Strategies and Practices in Medicinal Chemistry, 8 September 2011, Biopolis, Singapore.

17. 2’-Fluoro-4’-thioarabino-modified oligonucleotides: conformational switches linked to siRNA activity Watts Jonathan K., Choubdar Niloufar, Sadalapure Kashinath, Robert Francis, Wahba Alexander S., Pelletier Jerry, Pinto B. Mario and Damha Masad J. Nucleic Acids Research, 35 (5), 2007, 1441-1451.

18. Synthesis and conformational analysis of 2'-fluoro-5-methyl-4'-thioarabinouridine (4'S-FMAU) Watts, Jonathan K.; Sadalapure, Kashinath; Choubdar, Niloufar; Damha, Masad J.; Pinto, B. Mario. Abstracts of Papers, 231st ACS National Meeting, Atlanta, GA, United States, March 26-30, 2006, CARB-003.

19. Synthesis of functionalized amphiphilic glycoconjugates and glycoclusters Dubber, Michael; Patel, Anupama; Sadalapure, Kashinath; Aumueller, Ingo; Lindhorst, Thisbe K, Eur. J. Org Chem, 23, 2006, 5357-5366.

20. Synthesis and Conformational Analysis of 2'-Fluoro-5-methyl-4'-thio arabinouridine(4'S- FMAU). J. K. Watts, K. Sadalapure, N. Choubdar, B. Mario Pinto, and M. J. Damha J. Org. Chem., 71 (3), 2006, 921 –925.

21. Fluorescent Labelled Thiourea-bridged Glycodendrons. Krist Pavel; Vannucci Luca; Kuzma Marek; Man Petr; Sadalapure Kashinath; Patel Anupama Bezouska Karel; Pospisil Milan; Petrus Ladislav; Lindhorst Thisbe K.; Kren Vladimir ChemBioChem., 5 (4), 2004, 445-452.

22. Effects of N-acetyl-glucosamine-coated glycodendrimers as biological modulators in the B16F10 melanoma model in vivo. Vannucci Luca; Fiserova Anna; Sadalapure Kashinath; Lindhorst Thisbe K; Kuldova Marketa; Rossmann Pavel; Horvath Ondrej; Kren Vladimir; Krist Pavel; Bezouska Karel; Luptovcova Martina; Mosca Franco; Pospisil Miloslav, International J. Oncology, 23 (2), 2003, 285-296.

23. Glycodendrimeric ligands of C-type lectin receptors as therapeutic agents in experimental cancer. M. Pospisil; L. Vannucci; A. Fiserova; K. Krausova; O. Horvath; V. Kren; F. Mosca; Th. K. Lindhorst; K. S. Sadalapure; K. Bezouska, Adv. Exp. Med. Biol., 495, 2001, 343-347. A general entry in to glycopeptide dendrons, K. S. Sadalapure; Th. K. Lindhorst, Angew. Chem., Int. Ed. 39 (11), 2000, 2010-2013.

24. Glucose-based AB2-building blocks for the construction of branched glycopeptidomimetics C. Kieburg; K. S. Sadalapure; Th. K. Lindhorst, Eur. J. Org. Chem., 11, 2000, 2035-2040.

25. A carbohydrate route to CMI-977: a potent 5-lipoxygenase inhibitor. M. S. Chorghade; K. S. Sadalapure; S. Adhikari; SVS. Lalitha; AMS. Murugaiah; P. Radhakrishna; B. S. Reddy; M. K. Gurjar, Carbohydr. Lett., 3 (6), 2000, 405-410.

26. Synthesis of (2S, 5S)-trans-5-(4-fluorophenoxymethyl)-2- (1-N-hydroxyureidyl)-3-butyn-4-yl)-tetrahydrofuran (CMI-977) M. S. Chorghade; M. K. Gurjar; S. Adhikari; K. S. Sadalapure; SVS. Lalitha; AMS. Murugaiah; P. Radhakrishna, Pure and Appl. Chem., 71 (6), 1999, 1071-1074.

27. Synthesis and anomeric stability of (16)-thiourea-linked pseudo- oligosaccharides J. M. Benito; C. O. Mellet; K. S. Sadalapure; Th. K. Lindhorst; J. Defaye; J. M. G. Fernández, Carbohydr. Res., 320, 1999, 37-48.

28. Development of cost-effective syntheses of a potent 5-LO inhibitor M. S. Chorghade; M. K. Gurjar; K. S. Sadalapure; S. V. S. Lalitha; A. M. S. Murugaiah; P. Radhakrishna; S. Adhikari, Book of Abstracts, 216th ACS National Meeting, Boston, 1998, August 23rd –27th.

29. Kinetic resolution of aryl glycidyl ethers: a practical synthesis of optically pure -blocker, S-metoprolol M. K. Gurjar, K. S. Sadalapure, S. Adhikari, B. V. N. B. S. Sarma, M. S. Chorghade, Heterocycles, 48 (7), 1998, 1471-1476.

30. A practical synthesis of (R) and (S) -benzyl glycidols by hydrolytic kinetic resolution M. K. Gurjar; BVNBS. Sarma; K. S. Sadalapure; S. Adhikari, Synthesis, 10, 1998, 1424-1424.

31. Zaragozic acid : unusual stereochemical dependence in anhydride formation of carbohydrate templates M. K. Gurjar; S. K. Das; K. S. Sadalapure, Tetrahedron Lett., 36 (11), 1995, 1933-1936.

32. A Modular Approach for the Synthesis of Oligosaccharide Mimetics, Anupama Patel and Thisbe K. Lindhorst, J. Org. Chem. 2001, 66(8), 2674-2680.

33. Synthesis of "mixed type" oligosaccharide mimetics based on a carbohydrate scaffold. Anupama Patel and Thisbe K. Lindhorst, Eur. J. Org. Chem. 2002, 1, 79-89.

34. Efficient Synthesis of Isotopically Pure Isotope-Coded Affinity Tagging Reagents. Anupama Patel and David M. Perrin, Bioconjugate Chem. 2004, 15, 224-230.

35. Synthesis of functionalized amphiphilic glycoconjugates and glycoclusters. Dubber, Michael; Patel, Anupama; Sadalapure, Kashinath; Aumueller, Ingo; Lindhorst, Thisbe K, Eur. J. Org Chem, 23, 2006, 5357-5366.

36. Fluorescent Labelled Thiourea-bridged Glycodendrons.

37. Krist Pavel; Vannucci Luca; Kuzma Marek; Man Petr; Sadalapure Kashinath; Patel Anupama; Bezouska Karel; Pospisil Milan; Petrus Ladislav; Lindhorst Thisbe K.; Kren Vladimir ChemBioChem., 5 (4), 2004, 445-452.

38. Multivalent glycomimetics: synthesis of nonavalent mannoside clusters with variation of spacer properties. Anupama Patel and Thisbe K. Lindhorst; Carb.Res. 2006, 341(10), 1657-1668.

39. A mechanism-based proteomic strategy for monitoring cysteine proteases using cathepsin B-targeted ICAT reagents. Anupama Patel, Omid Hekmat, John S. Mort, Stephen G. Withers, and David M. Perrin. Unpublished work.

40. Synthesis of the C30-C38 fragment of the marine macrolide Altohyrtin, Anupama Patel and Mukund K. Gurjar. Unpublished work.